• litababjtp

"Bophelo ba nakong e fetileng le ba hona joale" ba berberine hydrochloride

Ho bua kaberberine , motho e mong le e mong e ka ’na eaba ha aa tloaeleha, empa e mong le e mong o tlameha ho tseba maele a tloaelehileng: Motho ea semumu o ja ma-coptis – a ke ke a bolela bohloko! Ke 'nete, karolo e ka sehloohong e babang ho coptis ke berberine, e leng berberine hydrochloride.

Berberine

Berberine (BBR) ke alkaloid ea isoquinoline - C20H19NO5 e ntšitsoeng ho Coptis chinensis. E fumaneha limeleng tsa meloko e 10 le malapa a 4 ho kenyeletsa le Berberidaceae. Likristale tse tšehla tse bōpehileng joaloka nale li ka tšeloa ho tloha diethyl ether, ka ntlha ea ho qhibiliha ea 145°C. Li qhibiliha ka metsing 'me ha li qhibilihe ka har'a benzene, diethyl ether le chloroform.

Lipatlisiso tsa morao-rao tsa meriana li tiisitse hore berberine e na le ho hloleha ho hoholo ha pelo, anti-arrhythmia, ho theola k'holeseterole, ho ata ha mesifa e thibelang methapo ea mali, ho ntlafatsa ho hanyetsa insulin, ho thibela-platelet, ho thibela ho ruruha le liphello tse ling. Ka hona, e ka ba molemo ho mafu a pelo le methapo ea methapo. Litebello tsa eona tse pharaletseng le tsa bohlokoa tsa tšebeliso li hohetse tlhokomelo e ntseng e eketseha. Ho ea ka lipatlisiso tsa morao-rao tsa bongaka, berberine e na le liphello tse ntle ho thibela le ho phekola khatello ea kelello, hyperlipidemia, lefu la tsoekere, arrhythmia, lihlahala le mafu a mang. Berberine hydrochloride e tlalehiloe haholo ka ho fokotsa lipids tsa mali. BBR e ka laola polelo ea "low-density lipoprotein receptor LDLR" le ho khothaletsa ho monngoa ha protheine ea LDL ke lisele tsa sebete. BBR e fetoloa dihydroberberine (dhBBR) ke nitroreductase ea mala a mala a microbiota, e etsa hore e monye habonolo ke mala. Ka mor'a ho monngoa, e kenngoa ka oxidized ho BBR ka har'a lisele tsa mala ebe e kena maling. Fumana litlamorao tsa ho theola lipid le hypoglycemic. BBR e ka boela ea ntlafatsa metabolism ea matla. Tsamaiso ea molomo ea BBR e khothalletsa gut microbiota ho hlahisa butyrate, e kenang maling 'me e sebetsa ho SCFAs (short chain fatty acids), e fokotsang lipids le maemo a tsoekere maling.

b4c363a2-2773-4e27-bd8a-8f89beef33aa_large BBR e ka khothaletsa nchafatso ea lisele tsa pancreatic islet mme e na le melemo e mengata ho feta litlhare tse ling tse thibelang lefu la tsoekere. Liteko tsa kliniki tse amehang li pakile hore berberine e ka thibela myocardial fibrosis ho likhoto tsa lefu la tsoekere; BBR e na le litlamorao tsa anti-platelet, e ka eketsa litaba tsa nucleotide ka har'a liplatelete le ho thibela ho kopana. Berberine e kopantsoe le li-statins e phetha karolo ea bohlokoa ho tsitsisa plasma trimethylamine oxidation ho lefu la pelo le ho thibela ho thehoa ha atherosclerosis.KHHEALTH10310458

Berberine ea Machaena ke mokhoa o mong o loketseng ho feta lithethefatsi tsa "statin". Kaha berberine e theko e tlase ka makhetlo a mangata ho feta lithethefatsi tsa "statins", ho sibolloa ha phello ea berberine ea ho theola lipid-lipid ho na le boleng bo sa lebelloang bakeng sa thibelo le kalafo ea hyperlipidemia, lefu la tsoekere le lefu la pelo.
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Nako ea poso: Jan-08-2024